Niacin

Niacin (Vitamin B3)
Also known as: Nicotinic acid, Vitamin B3
Vitamin & Mineral

Content by: OpenSupplement Editorial Team  |  Medical review: pending  |  Last updated: April 13, 2026

Supplement Score
Niacin500-2000 mg/day (extended-release) | $5-10/mo
Safety3
Interactions3
Cost5
Evid.Onset
Heart disease
33
2 PubMed references cited
4–5 Strong2–3 Emerging1 Weak|Methodology

TL;DR

  • Vitamin B3, used in high doses as a lipid-modifying medication

  • Moderate evidence for improving the 'cholesterol profile' (raises HDL)

  • Notable for causing the 'Niacin Flush' — an itchy, red skin reaction

  • Mixed results in recent large trials (AIM-HIGH, HPS2-THRIVE)

  • Cheap: ~$5-10/month

  • Best for: Low HDL cholesterol, high triglycerides

What it is

Niacin is an essential B vitamin involved in over 400 enzyme reactions. However, at 'mega-doses' (1,000mg+), it becomes a powerful drug for cholesterol. It was the primary lipid-lowering tool before statins were invented.

Niacin works by blocking the breakdown of fats in adipose tissue and the liver, which lowers triglycerides and raises 'good' HDL cholesterol. The 'flush' occurs because niacin triggers the release of prostaglandins that dilate the blood vessels in the skin.

What the research says

Relevance: Moderate
Typical dose: 500-2000 mg/day (extended-release)

Niacin's reputation has taken a hit recently. The Profile. It is the single most effective supplement for raising 'good' HDL cholesterol and lowering Lipoprotein(a). The Controversy. Large-scale trials (AIM-HIGH) showed that while Niacin improved cholesterol numbers, it didn't necessarily reduce heart attacks when added to a statin. Practical Use. It is still a valuable tool for those with very high triglycerides or those who cannot take statins. [1][2]

DISCLAIMER: The information provided on this page, including but not limited to text, graphics, images, and other material, is for informational and educational purposes only. No material is intended to be a substitute for professional medical advice, diagnosis, or treatment. Always seek the advice of your physician or other qualified healthcare provider with any questions you may have regarding a medical condition or treatment and before undertaking a new healthcare regimen. Never disregard professional medical advice or delay in seeking it because of something you have read on this website.

Use of this website does not create a doctor-patient relationship between you and OpenSupplement.org or its operators. Reliance on any information provided is solely at your own risk.

This page may contain affiliate links. If you purchase through these links, we may earn a small commission at no extra cost to you. Learn more.

Niacin on Amazon

$5-10/mo (estimated)
See on Amazon

Safety

High doses can be taxing on the liver; regular blood tests are recommended. The 'Niacin Flush' is harmless but uncomfortable. Avoid 'No-Flush' Niacin (Inositol Hexanicotinate), as it is generally ineffective for cholesterol. Extended-release (Slo-Niacin) is gentler but carries higher liver risk.

Interactions

  • Statins: May increase the risk of muscle pain (myopathy).
  • Diabetes Meds: High-dose niacin can raise blood sugar levels.
  • Gout: May increase uric acid levels, triggering gout attacks.

Dosing

For Cholesterol: 500-2,000 mg daily. Form: Immediate-release (for least liver risk) or Extended-release (for least flush). Tip: Take with a snack and an aspirin 30 minutes before to minimize flushing.

Cost

Very cheap. $5-10 per month.

The bottom line

Niacin is a powerful, old-school heart tool. It's not for everyone, but if you need to raise your HDL or lower triglycerides, it's the most effective 'vitamin' for the job.

References

  1. RCTHeart diseasePubMed
  2. NIH Fact SheetHeart diseaseSource

Sources for this page include published meta-analyses, systematic reviews, and NIH dietary supplement fact sheets. All claims reflect the evidence as of early 2026.

This is not medical advice. Consult your healthcare provider before starting any supplement, especially if you take medications.